Journal of Medicinal Chemistry
ISSNs: 0022-2623
American Chemical Society, United States
FI (2012): 2, ISI indexed (2012): yes
Central database
Journal
- 2013
- Published
Design, Synthesis, and Pharmacological Characterization of N- and O-Substituted 5,6,7,8-Tetrahydro-4H-isoxazolo[4,5-d]azepin-3-ol Analogues: Novel 5-HT2A/5-HT2C Receptor Agonists with Pro-Cognitive Properties. / Jensen, Anders A.; Plath, Niels; Pedersen, Martin Holst Friborg; Isberg, Vignir; Krall, Jacob; Wellendorph, Petrine; Stensbøl, Tine B.; Gloriam, David E.; Krogsgaard-Larsen, Povl; Frølund, Bente.
In: Journal of Medicinal Chemistry, Vol. 56, No. 3, 2013, p. 1211-1227.Publication: Research - peer-review › Journal article – Annual report year: 2013
- 2012
- Published
Disparate SAR Data of Griseofulvin Analogues for the Dermatophytes Trichophyton mentagrophytes, T. rubrum, and MDA-MB-231 Cancer Cells. / Rønnest, Mads Holger; Raab, Marc S.; Anderhub, Simon; Boesen, Sven; Krämer, Alwin; Larsen, Thomas Ostenfeld; Clausen, Mads Hartvig.
In: Journal of Medicinal Chemistry, Vol. 55, No. 2, 2012, p. 652-660.Publication: Research - peer-review › Journal article – Annual report year: 2012
- Published
Structure–Activity Relationship Study of Selective Excitatory Amino Acid Transporter Subtype 1 (EAAT1) Inhibitor 2-Amino-4-(4-methoxyphenyl)-7-(naphthalen-1-yl)-5-oxo-5,6,7,8-tetrahydro-4H-chromene-3-carbonitrile (UCPH-101) and Absolute Configurational Assignment Using Infrared and Vibrational Circular Dichroism Spectroscopy in Combination with ab Initio Hartree–Fock Calculations. / Huynh, Tri H.V.; Shim, Irene; Bohr, Henrik; Abrahamsen, Bjarke; Nielsen, Birgitte; Jensen, Anders A.; Bunch, Lennart.
In: Journal of Medicinal Chemistry, Vol. 55, No. 11, 2012, p. 5403-5412.Publication: Research - peer-review › Journal article – Annual report year: 2012
- Published
Substrates for Efficient Fluorometric Screening Employing the NAD-Dependent Sirtuin 5 Lysine Deacylase (KDAC) Enzyme. / Madsen, Andreas Stahl; Olsen, Christian Adam.
In: Journal of Medicinal Chemistry, Vol. 55, No. 11, 2012, p. 5582-5590.Publication: Research - peer-review › Journal article – Annual report year: 2012
- 2010
- Published
Design, Synthesis, and in Vitro Pharmacology of New Radiolabeled γ-Hydroxybutyric Acid Analogues Including Photolabile Analogues with Irreversible Binding to the High-Affinity γ-Hydroxybutyric Acid Binding Sites. / Sabbatini, Paola; Wellendorph, Petrine; Høg, Signe; Pedersen, Martin Holst Friborg; Bruner-Osborne, Hans; Martiny, Lars; Frølund, Bente; Clausen, Rasmus P.
In: Journal of Medicinal Chemistry, Vol. 53, No. 17, 2010, p. 6506-6510.Publication: Research - peer-review › Journal article – Annual report year: 2010
- Published
Liposomal Formulation of Retinoids Designed for Enzyme Triggered Release. / Pedersen, Palle Jacob; Adolph, Sidsel Kramshøj; Subramanian, Arun Kumar; Arouri, A.; Andresen, Thomas Lars; Mouritsen, O.G.; Madsen, Robert; Madsen, M.W.; Peters, Günther H.J.; Clausen, Mads Hartvig.
In: Journal of Medicinal Chemistry, Vol. 53, No. 9, 2010, p. 3782-3792.Publication: Research - peer-review › Journal article – Annual report year: 2010
- 2009
- Published
Synthesis and Biophysical Characterization of Chlorambucil Anticancer Ether Lipid Prodrugs. / Pedersen, Palle Jacob; Christensen, Mikkel Stochkendahl; Ruysschaert, Tristan; Linderoth, Lars; Andresen, Thomas Lars; Melander, Fredrik; Mouritsen, Ole G.; Madsen, Robert; Clausen, Mads Hartvig.
In: Journal of Medicinal Chemistry, Vol. 52, No. 10, 2009, p. 3408-3415.Publication: Research - peer-review › Journal article – Annual report year: 2009
- Published
Synthesis and Structure-Activity Relationship of Griseofulvin Analogues as Inhibitors of Centrosomal Clustering in Cancer Cells. / Rønnest, Mads Holger; Rebacz, Blanka; Markworth, Lene; Terp, Anette Hinsch; Larsen, Thomas Ostenfeld; Krämer, A.; Clausen, Mads Hartvig.
In: Journal of Medicinal Chemistry, Vol. 52, No. 10, 2009, p. 3342-3347.Publication: Research - peer-review › Journal article – Annual report year: 2009
- 2007
- Published
In silico prediction of cytochrome P450 2D6 and 3A4 inhibition using Gaussian kernel weighted k-nearest neighbor and extended connectivity fingerprints, including structural fragment analysis of inhibitors versus noninhibitors. / Jensen, B.F.; Vind, C.; Padkjær, S.B.; Brockhoff, Per B.; Refsgaard, H.H.
In: Journal of Medicinal Chemistry, Vol. 50, No. 3, 2007, p. 501-511.Publication: Research - peer-review › Journal article – Annual report year: 2007
- Submitted
Quantitative Modeling of Selective Lysosomal Targeting by Passive Diffusion of Xenobiotic Compounds : Model Development and Simulations for Single Cells. / Trapp, Stefan; Rosania, Gus; Horobin, Richard W. ; Kornhuber, Johannes.
In: The Journal of Medicinal Chemistry, 2007.Publication: Research › Journal article – Annual report year: 2007